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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T8239 Cromoglicic acid

Others Others
Cromoglicic acid 可防止肥大细胞释放炎性化学物质,例如组胺。
T0211 Azelastine

Azelastina,Astelin,Azelastinum,氮卓斯汀

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine (Azelastinum) 是一种选择性组胺 1 拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T3979 Emedastine

LY188695,依美斯汀,Emadine

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Emedastine (LY188695) 是一种可口服的,选择性和高亲和力的组胺 H1受体拮抗剂,Ki 值为 1.3 nM。它是苯并咪唑衍生物,可用于过敏性鼻炎、过敏性皮肤疾病和过敏性结膜炎的研究。
T0118 Mizolastine

SL 850324,咪唑司汀,咪唑斯汀

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mizolastine (SL 850324) 是组胺 H1 受体拮抗剂,IC50为 47 nM。它用于治疗过敏反应,如花粉热和荨麻疹等。
T21404 Fluticasone furoate

Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate

Glucocorticoid Receptor Endocrinology/Hormones
Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇,衍生自氟替卡松,Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。
T6242 Rupatadine Fumarate

富马酸卢帕他定,Rinialer,Rupafin,Alergoliber

PAFR; Autophagy; Histamine Receptor Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Rupatadine Fumarate (Rinialer) 是一种可口服的长效PAF/H1受体的双抑制剂,Ki 值分别为 0.55 μM 和 0.1 μM。它可研究过敏性鼻炎和荨麻疹。
T0059 Diphenylpyraline hydrochloride

盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂,抑制多巴胺的吸收。它是可口服的抗组胺试剂,具有抗胆碱和抗过敏作用,可用于缓解过敏性疾病,如鼻炎、花粉热和瘙痒性皮肤疾病等。
T3185 R112

(E)-Elafibranor

Syk Angiogenesis; Tyrosine Kinase/Adaptors
R112 ((E)-Elafibranor) 是ATP 竞争性的 Syk 激酶抑制剂,它能够抑制Syk 激酶活性,Ki=6 nM,IC50=226 nM。
T0211L Azelastine hydrochloride

Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine hydrochloride (Astelin) 是一种选择性组胺 1拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T1030 Triprolidine hydrochloride monohydrate

盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Triprolidine hydrochloride monohydrate 是一种组胺 H1 拮抗剂,用于过敏性鼻炎、哮喘。
T1269 Tripelennamine hydrochloride

Pyribenzamine hydrochloride,去敏灵,Tripelennamine HCl,Pyribenzamine HCl,盐酸曲吡那敏

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) 是一种组胺 H1 拮抗剂,具有低镇静作用,但经常刺激胃肠道。
T2335 Ebastine

Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ebastine (Kestine) 是一种可口服的组胺 H1 受体拮抗剂,用于过敏性鼻炎的症状和慢性特发性荨麻疹的研究。
T0188 Fluticasone (propionate)

丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate

Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Microbiology/Virology
Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,亲和力KD 为 0.5 nM。具有抗病毒活性。
T0205 Brompheniramine maleate

Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Brompheniramine maleate (Dimotane) 是一种可口服的丙胺类抗组胺剂,具有抗胆碱能和抗抑郁作用,可用于过敏性鼻炎和缓解疼痛的研究。它是一种选择性组胺 H1 受体拮抗剂,Kd 为 6.06 nM。
T0089 Cetirizine dihydrochloride

盐酸西替利嗪,P071,UCB P071,Cetirizine DiHCl

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Cetirizine dihydrochloride (UCB P071) 是羟嗪的羧化代谢物,是特异性口服有效的 H1 受体长效拮抗剂。它标记抗过敏特性,抑制过敏反应期间嗜酸性粒细胞趋化,可有效治疗过敏性鼻炎、确诊荨麻疹和花粉诱发的哮喘。
T6660 SB-705498

TRP/TRPV Channel Membrane transporter/Ion channel
SB705498 是一种口服有效的 TRPV1选择性拮抗剂,pIC50值为 7.1。
T1553 Chlorpheniramine maleate

马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Chlorpheniramine maleate (NCI-C55265) 是一种组胺 H1 拮抗剂,IC50为12 nM,用于过敏反应、花粉热、鼻炎、荨麻疹和哮喘。
T1531 Mometasone furoate

糠酸莫美他松,糠酸莫米松,Sch32088

Glucocorticoid Receptor Endocrinology/Hormones
Mometasone furoate (Sch32088) 是糖皮质激素受体激动剂,具有抗炎和抗过敏作用。它是皮质固醇类试剂,动物模型中,可局部应用于气道炎症、慢性皮肤湿疹、哮喘。
T2270 Trans-Tranilast

Tranilast trans-,反式-曲尼司特,反-曲尼司特

RAAS Endocrinology/Hormones
Trans-Tranilast 是抗过敏剂,可用于过敏性鼻炎、支气管哮喘和特应性皮炎的研究。
T1278 Astemizole

Laridal,Histaminos,Paralergin,阿司咪唑

Potassium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Astemizole (Laridal) 是一种长效、非镇静抗组胺药,用于治疗季节性过敏性鼻炎、哮喘、过敏性结膜炎和慢性特发性荨麻疹。它是组胺 H1 受体的拮抗剂,IC50值为 4 nM,还阻断 hERG K+通道,IC50值为 0.9 nM,具有抗胆碱能和止痒作用。
T2396 Ramatroban

BAY u3405,雷马曲班

GPR; Prostaglandin Receptor; PPAR DNA Damage/DNA Repair; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism
Ramatroban (BAY u3405) 是一种血栓素 A(2) (TxA(2)) 拮抗剂,IC50为 14 nM。它还通过抑制PGD2结合从而拮抗CRTH2,IC50为113 nM。它用于治疗过敏性鼻炎,可用于治疗哮喘的研究。
T77426 Pascolizumab

SB-240683

IL Receptor Immunology/Inflammation
Pascolizumab (SB-240683) 是一种人源化抗 IL-4 单克隆抗体。Pascolizumab 具有哮喘作用,可用于研究过敏性鼻炎。
T1470 Fexofenadine hydrochloride

Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,盐酸非索非那定,Telfast,Fexofenadine HCl,Allegra,MDL 16455A

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) 是一种抗组胺药,用于治疗过敏性鼻炎、血管性水肿和慢性荨麻疹。
T22354 Levocetirizine Dihydrochloride

Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydrochloride is the R-enantiomer of Cetirizine, which gives it a higher affinity for the H1-receptor than the S-enantiomer. Due to this enhanced affinity, Levocetirizine Dihydrochloride is effective in treating allergic rhinitis and chronic idiopathic urticaria.
T1097 Loratadine

氯雷他定,SCH 29851,Loratidine

Influenza Virus; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Loratadine (SCH 29851) 是一种组胺 H1受体反向激动剂,IC50>32 μM。它抑制炎症介质的免疫释放,具有抗登革热病毒的活性。
T61213 PF-03654764

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
PF-03654764 是一种具有口服活性、高效性和选择性的组胺 H3 受体拮抗剂,对人 H3 和大鼠 H3 具有抑制作用, Ki 值分别为 1.2 nM 和 7.9 nM。PF-03654764 常与 Fexofenadine 一起联合用药来治疗过敏性鼻炎。
T2392 Nafamostat mesylate

甲磺酸萘莫司他,FUT-175

Apoptosis; Serine/threonin kinase; SARS-CoV; Serine Protease Apoptosis; Cell Cycle/Checkpoint; Metabolism; Microbiology/Virology; Proteases/Proteasome
Nafamostat mesylate (FUT-175) 是一种广谱丝氨酸蛋白酶抑制剂,血管舒缓素抑制剂,能抑制血液凝固。它通过降低颗粒酶活性和 CTL 细胞溶解抑制T 细胞自身反应活性,可抑制SARS-CoV-2 的激活。它还是潜在的补体抑制剂。
T4563 Thonzylamine

neohetramine,松齐拉敏

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Thonzylamine (neohetramine) 是可口服的H1组胺受体拮抗剂,具有抗组胺和抗过敏特性,可用于鼻充血、过敏性结膜炎和其他过敏性疾病的研究。
T21112 Triprolidine hydrochloride

295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil

Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.
T10437 AZD8848

TLR Immunology/Inflammation
AZD8848 is a selective antedrug agonist of toll-like receptor 7 (TLR7). It is developed for the research of asthma and allergic rhinitis.
T69737 SCH-79687

SCH-79687 is a histamine antagonist selective for the H3 subtype. This H3 antagonist may play a role in allergic rhinitis.
T29951 Ambicromil

Ambicromil is used for allergic rhinitis.
T0785L Dexchlorpheniramine free base

Polaramine,Dexchlorpheniramine Maleate,Mylaramine

Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.
T27556 HSR-609

HSR609,FY609,FY-609,FY 609

HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.
T27445 GSK-1004723

GSK 1004723

GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.
T37386 Dihydro Montelukast

Dihydro montelukast is a potential impurity found in commercial montelukast preparations. Montelukast (sodium salt) is a potent and selective cysteinyl leukotriene 1 (CysLT1) receptor antagonist. Formulations containing montelukast are used for the treatment of asthma as well as for the symptoms associated with allergic rhinitis.
T21247 Carbinoxamine

Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine

Carbinoxamine, an anticholinergic and antihistamine agent, is used for hay fever, angioedema, vasomotor rhinitis, mild urticaria, dermatographism and allergic conjunctivitis. It is a histamine antagonist, specifically an H1-antagonist.
T74646 PM-81I

PM-81I为一种高效STAT6抑制剂(针对SH2结构域),可显著减少STAT6的磷酸化水平。适用于研究过敏性肺病、过敏性鼻炎、慢性阻塞性肺病或癌症。
T26770 Bencycloquidium Bromide

BCQB

Bencycloquidium Bromide is a muscarinic M3 antagonist. Bencycloquidium bromide inhibits nasal hypersecretion in a rat model of allergic rhinitis. Bencycloquidium Bromide showed high affinity toward the M(3) receptor in Chinese hamster ovary (CHO) cells (M
T16476 PF-03654746

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。
T73972 Fexofenadine Impurity F

Fexofenadine Impurity F 是 Fexofenadine 的杂质。 Fexofenadine 是一种H1R 拮抗剂,可用于研究季节性过敏性鼻炎和慢性特发性荨麻疹。
T60514 Triprolidine

Triprolidine 是一种口服活性的组胺H1受体拮抗剂,可用于过敏性鼻炎的研究 。Triprolidine 具有脊髓运动和知觉阻止的作用。
T62669 Tripelennamine citrate

Tripelennamine citrate 是一种乙二胺衍生物,是一种有效的组胺 H1 受体拮抗剂。Tripelennamine citrate 能够减少组织胺引起的机体过敏反应。Tripelennamine citrate 能够用于研究鼻炎、结膜炎、过敏性和过敏性反应。
T73129 STAT6-IN-1

STAT6-IN-1(化合物19a)是一种针对STAT6的SH2结构域表现出较高亲和力(IC50=0.028 µM)的STAT6抑制剂。该化合物主要用于研究过敏性肺病、过敏性鼻炎、慢性阻塞性肺病或癌症。
T60392 Tripelennamine

Tripelennamine 是一种乙二胺衍生物,是一种有效的组胺 H1受体拮抗剂,可减轻由组织胺引起的机体过敏反应。Tripelennamine 可用于鼻炎、结膜炎、过敏性和过敏性反应的研究。
T68280 Adriforant

Adriforant, also known as ZPL-3893787, PF-3893787 and ZPL-389, is a novel histamine H4 receptor antagonist. Adriforant shows an excellent in vitro profile that warrants their further investigation in relevant models of human disease. Histamine H4 receptor (H4R) has become a promising target for immuno-inflammatory diseases, such as allergic rhinitis, asthma or dermal allergies.
T38350 TAS 205

TAS 205 is an inhibitor of hematopoietic prostaglandin D synthase (H-PGDS; IC50= 55.8 nM).1It is selective for H-PGDS over lipocalin-type PGDS (L-PGDS) at 100 μM, as well as over enzyme and receptor panels at 10 μM. TAS 205 inhibits production of prostaglandin D2induced by A23187 in KU812 human and RBL-2H3 rat basophils with IC50values of 78.3 and 181.3 nM, respectively. It inhibits ovalbumin-induced nasal lavage fluid eosinophil infiltration and late-phase nasal obstruction in an ovalbumin-sens...
T69918 Adriforant tartrate hydrate

Adriforant, also known as ZPL-3893787, PF-3893787 and ZPL-389, is a novel histamine H4 receptor antagonist. Adriforant shows an excellent in vitro profile that warrants their further investigation in relevant models of human disease. Histamine H4 receptor (H4R) has become a promising target for immuno-inflammatory diseases, such as allergic rhinitis, asthma or dermal allergies.
T60843 Brompheniramine

Brompheniramine ((±)-Brompheniramine) 是具有口服活性的烷基胺类抗组胺药。Brompheniramine 是组胺 H1 受体的选择性拮抗剂 (Kd = 6.06 nM)。Brompheniramine 可用于过敏性鼻炎,它具有抗胆碱能、抗抑郁和麻醉作用。Brompheniramine 可阻断钙离子通道、钠离子通道和 hERG 通道,IC50分别为 16.12 μM, 21.26 μM 和 0.90 μM。
T74583 Desmethylazelastine

Desmethylazelastine是Azelastine经由细胞色素P450酶系统的氧化代谢形成的主要活性代谢物,具有97%的蛋白结合率和54小时的消除半衰期。Azelastine作为一种口服活性的组胺H1受体拮抗剂,特点是选择性高和亲和力强。它主要用于治疗过敏性鼻炎、哮喘、糖尿病高脂血症以及用于SARS-CoV-2的研究。

化合物

Cromoglicic acid
Cat.No: T8239
Synonym:
Target: Others
Azelastine
Cat.No: T0211
Synonym: Azelastina,Astelin,Azelastinum,氮卓斯汀
Target: SARS-CoV, Histamine Receptor
Emedastine
Cat.No: T3979
Synonym: LY188695,依美斯汀,Emadine
Target: Histamine Receptor
Mizolastine
Cat.No: T0118
Synonym: SL 850324,咪唑司汀,咪唑斯汀
Target: Histamine Receptor
Fluticasone furoate
Cat.No: T21404
Synonym: Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate
Target: Glucocorticoid Receptor
Rupatadine Fumarate
Cat.No: T6242
Synonym: 富马酸卢帕他定,Rinialer,Rupafin,Alergoliber
Target: PAFR, Autophagy, Histamine Receptor
Diphenylpyraline hydrochloride
Cat.No: T0059
Synonym: 盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride
Target: Histamine Receptor
R112
Cat.No: T3185
Synonym: (E)-Elafibranor
Target: Syk
Azelastine hydrochloride
Cat.No: T0211L
Synonym: Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin
Target: SARS-CoV, Histamine Receptor
Triprolidine hydrochloride monohydrate
Cat.No: T1030
Synonym: 盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride
Target: Histamine Receptor
Tripelennamine hydrochloride
Cat.No: T1269
Synonym: Pyribenzamine hydrochloride,去敏灵,Tripelennamine HCl,Pyribenzamine HCl,盐酸曲吡那敏
Target: Histamine Receptor
Ebastine
Cat.No: T2335
Synonym: Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305
Target: Histamine Receptor
Fluticasone (propionate)
Cat.No: T0188
Synonym: 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate
Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite
Brompheniramine maleate
Cat.No: T0205
Synonym: Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane
Target: 5-HT Receptor, Histamine Receptor
Cetirizine dihydrochloride
Cat.No: T0089
Synonym: 盐酸西替利嗪,P071,UCB P071,Cetirizine DiHCl
Target: Histamine Receptor
SB-705498
Cat.No: T6660
Synonym:
Target: TRP/TRPV Channel
Chlorpheniramine maleate
Cat.No: T1553
Synonym: 马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate
Target: Histamine Receptor
Mometasone furoate
Cat.No: T1531
Synonym: 糠酸莫美他松,糠酸莫米松,Sch32088
Target: Glucocorticoid Receptor
Trans-Tranilast
Cat.No: T2270
Synonym: Tranilast trans-,反式-曲尼司特,反-曲尼司特
Target: RAAS
Astemizole
Cat.No: T1278
Synonym: Laridal,Histaminos,Paralergin,阿司咪唑
Target: Potassium Channel, Histamine Receptor
Ramatroban
Cat.No: T2396
Synonym: BAY u3405,雷马曲班
Target: GPR, Prostaglandin Receptor, PPAR
Pascolizumab
Cat.No: T77426
Synonym: SB-240683
Target: IL Receptor
Fexofenadine hydrochloride
Cat.No: T1470
Synonym: Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,盐酸非索非那定,Telfast,Fexofenadine HCl,Allegra,MDL 16455A
Target: Histamine Receptor
Levocetirizine Dihydrochloride
Cat.No: T22354
Synonym: Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride
Target: Histamine Receptor
Loratadine
Cat.No: T1097
Synonym: 氯雷他定,SCH 29851,Loratidine
Target: Influenza Virus, Histamine Receptor
PF-03654764
Cat.No: T61213
Synonym:
Target: Histamine Receptor
Nafamostat mesylate
Cat.No: T2392
Synonym: 甲磺酸萘莫司他,FUT-175
Target: Apoptosis, Serine/threonin kinase, SARS-CoV, Serine Protease
Thonzylamine
Cat.No: T4563
Synonym: neohetramine,松齐拉敏
Target: Histamine Receptor
Triprolidine hydrochloride
Cat.No: T21112
Synonym: 295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil
Target:
AZD8848
Cat.No: T10437
Synonym:
Target: TLR
SCH-79687
Cat.No: T69737
Synonym:
Target:
Ambicromil
Cat.No: T29951
Synonym:
Target:
Dexchlorpheniramine free base
Cat.No: T0785L
Synonym: Polaramine,Dexchlorpheniramine Maleate,Mylaramine
Target:
HSR-609
Cat.No: T27556
Synonym: HSR609,FY609,FY-609,FY 609
Target:
GSK-1004723
Cat.No: T27445
Synonym: GSK 1004723
Target:
Dihydro Montelukast
Cat.No: T37386
Synonym:
Target:
Carbinoxamine
Cat.No: T21247
Synonym: Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine
Target:
PM-81I
Cat.No: T74646
Synonym:
Target:
Bencycloquidium Bromide
Cat.No: T26770
Synonym: BCQB
Target:
PF-03654746
Cat.No: T16476
Synonym:
Target: Histamine Receptor
Fexofenadine Impurity F
Cat.No: T73972
Synonym:
Target:
Triprolidine
Cat.No: T60514
Synonym:
Target:
Tripelennamine citrate
Cat.No: T62669
Synonym:
Target:
STAT6-IN-1
Cat.No: T73129
Synonym:
Target:
Tripelennamine
Cat.No: T60392
Synonym:
Target:
Adriforant
Cat.No: T68280
Synonym:
Target:
TAS 205
Cat.No: T38350
Synonym:
Target:
Adriforant tartrate hydrate
Cat.No: T69918
Synonym:
Target:
Brompheniramine
Cat.No: T60843
Synonym:
Target:
Desmethylazelastine
Cat.No: T74583
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S0878 Prunetin

樱黄素,Prunusetin

ERK; Dehydrogenase; NF-κB MAPK; Metabolism; NF-κB
Prunetin (Prunusetin) 是一种O-甲基化异黄酮,具有抗炎的作用。它是人醛脱氢酶的有效抑制剂。
T4038 Ectoine

THP(B),L-Ectoine,四氢甲基嘧啶羧酸

Others; Antibacterial Microbiology/Virology; Others
Ectoine (L-Ectoine) 是生活在极其恶劣环境中的细菌所产生的氨基酸衍生物,是一种天然的细胞保护剂。它具有良好的安全性,可研究过敏性鼻炎。它用作渗透调节相容性溶质,可增加皮肤表面的水合作用并稳定脂质层,常用于皮肤护理。

天然产物

Prunetin
Cat.No: T4S0878
Synonym: 樱黄素,Prunusetin
Target: ERK, Dehydrogenase, NF-κB
Ectoine
Cat.No: T4038
Synonym: THP(B),L-Ectoine,四氢甲基嘧啶羧酸
Target: Others, Antibacterial
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